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  1. Pubblicazioni

IL FARMACO

Rivista
Codice:
E062766
ISSN:
0014-827X
  • Dati Generali

Dati Generali

Pubblicazioni (84)

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1,2,3-triazolo 4,5-f quinolines. II. Preparation and antimicrobial evaluation of 6-ethyl-6,9-dihydro-1(2)(3)-R-1(2)(3)H-triazolo 4,5-f quinolin-9-one-8-carboxylic acids as anti-infectives of the urinary tract (1)
Articolo
1,2,3-triazolo[4,5-f]quinolines: II: preparation and antimicrobial evaluation of 6-ethyl-6,9-dihydro-1(2)(3)-R-1(2) (3)H-triazolo [4,5-f]quinolin-9-one-8-carboxylic acids as anti-infectives of the urinary tract
Articolo
1,2,3-triazolo[4,5-h]quinolines. III. Preparation and antimicrobial evaluation of 4-ethyl-4,7-dihydro-1(2)-R-1(2)H triazolo[4,5-h]quinolin-7-one-6-carboxylic acids as anti-infectives of the urinary tract.
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1,2,3-triazolo[4,5-h]quinolines: III: preparation and antimicrobial evaluation of 4-ethyl-4,7-dihydro-1(2)-R-1(2)H triazolo[4,5-h]quinolin-7-one-6-carboxylic acids as anti-infectives of the urinary tract
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1,4-Disubstituted 1,3-dihydro-2H-1,5-benzo- and chlorobenzodiazepin-2-ones with activity on the central nervous system (CNS)
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Amides and formamidines with antinociceptive activity (Note I)
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Amides and formamidines with antinociceptive activity (Note II)
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Amides and formamidines with antinociceptive activity: note I
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Amides and formamidines with antinociceptive activity: note II
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Antispasmodic activity of tert-aminoalkylderivatives of 3-benzyl-, 3-benzylaza- and 3-benzyldiazaquinoxalinones
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Benzocondensed derivatives as rigid analogues of the mu-opioid agonist 3(8)-cinnamyl-8(3)-propionyl-3,8-diazabicyclo[3.2.1]octanes: synthesis, modeling, and affinity
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Cellulose polymers for the constant release of a water-insoluble benzodiazepine
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Choleretic activity of 3-[ring substituted benzotriazol-1(2)-yl] alkanoic and alkenoic acids
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Chromophore-modified bis-benzo[g]indazole carboxamides: synthesis and antiproliferactive activity of bis-benzo[g]indazole carboxamides and related dimers
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Cyclopentenyl ethylamines active on CNS
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Cyclopentenyl ethylamines active on CNS
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DIURETIC AGENTS RELATED TO INDAPAMIDE .3. SYNTHESIS AND PHARMACOLOGICAL ACTIVITY OF N-(4-CHLORO-3-SULFAMOYLBENZAMIDO)-1,2,3,4-TETRAHYDROQUINOLINES AND 1,2,3,4-TETRAHYDROISOQUINOLINES
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DIURETIC AGENTS RELATED TO INDAPAMIDE .4. SYNTHESIS AND PHARMACOLOGICAL ACTIVITY OF N-(4-CHLORO-3-SULFAMOYLBENZAMIDO)-METHYL-PHENYL-PYRROLIDINES AND N1-(4-CHLORO-3-SULFAMOYLBENZOYL)-N2-ARYL OR ARALKYL-ALKYL-HYDRAZINES
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Diuretic agents related to indapamide. III--Synthesis and pharmacological activity of N-(4-chloro-3-sulfamoylbenzamido)-1,2,3,4-tetrahydroquinolines and 1,2,3,4-tetrahydroisoquinolines.
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Formamidines with antinociceptive and antiinflammatory activities
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Formamidines with antinociceptive and antiinflammatory activities
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Fungicidal Activity of Some o-nitrophenyl-hydrazones
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Fungicidal activity of some o-nitrophenil-hidrazones
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Fungicidal activity of some o-nitrophenyl-hydrazones
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Gold(I) complexes as antimicrobial agents
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Isolation, Characterization and Pharmacological Activity of Magydaris Pastinaca (LAM) Paol. Glucosides
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Isolation, characterization and pharmacological activity of Magydaris pastinacea Lam. Paol. glucosides
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Isolation, characterization and pharmacological activity ofMagydaris pastinacea(Lam.) Paol.glucosides
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Novel functionalized pyrido[2,3-g]quinoxalinones as antibacterial, antifungal and anticancer agents
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Preparation and biological evaluation of 6/7-trifluoromethyl(nitro)-, 6,7-difluoro-3-alkyl (aryl)-substituted-quinoxalin-2-ones. Part 3
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Pyridazine N-oxides .1. Synthesis and in vitro antimicrobial evaluation of 3-methyl-4-aryl-6-R-pyridazine N-oxides
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Pyridazine N-oxides .2. Synthesis and in vitro antimicrobial evaluation of 3-chloro-4-carbamoyl-5-aryl-6-methyl-pyridazine N-oxides
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Pyridazine N-oxides. I. Synthesis and in vitro antimicrobial evaluation of 3-methyl-4-aryl-6-R-pyridazine N-oxides
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Pyridazine N-oxides. II. Synthesis and in vitro antimicrobial evaluation of 3-chloro-4-carbamoyl-5-aryl-6-methyl-pyridazine N-oxides
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Quinoxalin-2-ones. Part 5. Synthesis and antimicrobial evaluation of 3-alkyl-, 3-halomethyl- and 3-carboxyethylquinoxaline-2-ones variously substituted on the benzo-moiety
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Quinoxaline Chemistry Part 12. 3-Carboxy-2[phenoxy]-6(7)substituted quinoxaline and N-[4-(6(7)substituted-3-carboxyquinoxalin-2-yl)hydroxy]benzoylglutamates. Synthesis and evaluation of in vitro anticancer activity
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Quinoxaline Chemistry. Part 17. 4[3,6(7) disubstituted-2-quinoxalinyl-oxa]phenylacetate and phenylacetylglutamate analogues of methotrexate: Synthesis and evaluation of in vitro anticancer activity
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Quinoxaline chemistry Part.10 Quinoxaline 10-oxa-analogues of trimetrexate (TMQ) and of 5,8-dideazafolic acid. Synthesis and evaluation of in vitro anticancer activity
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Quinoxaline chemistry. Part 8. 2-[Anilino]-3-[carboxy]-6(7)-substituted quinoxalines as non classical antifolate agents. Synthesis and evaluation of in vitro anticancer, anti-HIV and antifungal activity
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Quinoxaline chemistry. Part 13: 3-carboxy-2-benzylamino-substituted quinoxaline and N-[4-[(3-carboxyquinoxalin-2-yl)aminomethyl]benzoyl]-L-glutamates: synthesis and evaluation of in vitro anticancer activity
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Quinoxaline chemistry. Part 14. 4-(2-quinoxalylamino)-phenylacetates and 4-(2-quinoxalylamino)-phenylacetyl-L-glutamates as analogues-homologues of classical antifolate agents. Synthesis and evaluation of in vitro anticancer activity
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Quinoxaline chemistry. Part 15.4-[2-quinoxalylmethylenimino]-benzoylglutamates and benzoates, 4-[2-quinoxalylmethyl-N-methylamino]-benzoylglutamates as analogues of classical antifolate agents. Synthesis, elucidation of structures and in vitro evaluation of antifolate and anticancer activities
Articolo
Quinoxaline chemistry. Part 16. 4-Substituted anilino and 4-substituted phenoxymethyl pyrrolo[1,2-a]quinoxalines and N-[4-(pyrrolo[1,2-a]quinoxalin-4-yl)amino and hydroxymethyl]benzoyl glutamates. Symthesis and evaluation of in vitro biological activity
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Quinoxaline chemistry. Part 6- Synthesis and evaluation of antiulcer and gastroprotective activity of 2 –[arylmethylmercapto- arylmethylsulfinyl- piperazinyl- 3- r- substitute] quinoxalines.
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Quinoxaline chemistry. Part 8. 2-[anilino]-3- [carboxy]-6(7)-substituted quinoxalines as non classical antifolate agents. Synthesis and evaluation of in vitro anticancer, anti-HIV and antifungal activity
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Quinoxaline chemistry. Part11. 3-Phenyl-2-[phenoxy-and phenoxymethyl]-6(7) or 6,8-substituted quinoxalines and N-[4-(6(7)-substituted or 6,8-disubstituted-3-phenylquinoxalin-2-yl)hydroxy or hydroxymethyl]benzoylglutamates. Synthesis and evaluation of in vitro anticancer activity and enzymatic inhibitory activity against dihydrofolate reductase and thymidylate synthase
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Quinoxaline chemistry.Part 6 Synthesis and evaluation of antiulcer and gastroproctetive activity of 2-[arylmethylmercapto-,arylmethylsulfinyl-,piperazinyl-3-R-substituted]quinoxalines
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SYNTHESIS AND PHARMACOLOGICAL ACTIVITY OF 4-CARBAMOYL-6-BETA-THIENYL-4,5-DIHYDROPYRIDAZIN-3-(2H)ONES
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SYNTHESIS AND PHARMACOLOGICAL STUDY OF 4,4A,5,6-TETRAHYDRO-4A-SUBSTITUTED-BENZO(H)CINNOLIN-3(2H)ONES
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Sinthesis and evaluation of gastroproctetive activity of omeprazole related benzimidazole,imidazo[4,5-b]pyridine and quinoxaline 2-substituted derivatives
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Synthesis and CNS activities of pyridopyrazinone and pyridodiazepinone derivatives
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Synthesis and CNS activities of pyridopyrazinones and pyridodiazepinones derivatives
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Synthesis and D-2-like binding affinity of 4,5-dihydro-1H-benzo[g]indole-3-carboxamide derivatives as conformationally restricted 5-phenyl-pyrrole-3-carboxamide analogs
Articolo
Synthesis and antiinflammatory activity of some imidazolinyl - pyrazole derivatives
Articolo
Synthesis and antimycobacterial activity of 3-aryl-, 3-cyclohexyl- and 3-heteroaryl- substituted-2-(1H(2H)-benzotriazol-1(2)-yl)prop-2-enenitriles, prop-2-enamides and propenoic acids. II
Articolo
Synthesis and antiproliferative activity of 3-aryl-2-[1H(2H)-benzotriazol-1(2)-yl]acrylonitriles variously substituted: Part 4
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Synthesis and choleretic activity of 3-[2-(3-R', 4-R'', 5-R'''-benzyl)-5-R-benzimidazol-1-yl]-butanoic acids
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Synthesis and choleretic activity of 3-[2-(3-R', 4-R'', 5R'''-Benzyl)-5-R-Benzimidazol-1-YL]- Butanoic acids
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Synthesis and cytotoxicity evaluation of thiophene analogues of 1-methyl-2,3-bis(hydroxymethyl)benzo[g]indole bis[N-(2-propyl)carbamate]
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Synthesis and dopamine D2-like receptor binding affinity of substituted 5-phenyl-pyrrole-3-carboxamides
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Synthesis and evaluation for biological actvity of 3-alkyl and 3-halogenoalkyl-quinoxalin-2-ones variously substituted. Part 4
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Synthesis and evaluation of gastroprotective and antiulcer activity of some 2- substituted-1H-imidazo[4,5-b] pyridines and -1H-benzimidazoles
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Synthesis and evaluation of gastroprotective and antiulcer of some 2-substituted- 1H- imidazo[4,5-b]pyridines and 1H- benzimidazoles.
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Synthesis and in vitro anticancer activity evaluation of biscarbamic esters of 2,3-bis(hydroxymethyl)-1-methyl-7- and 7,8-substituted- benzo[g]indoles
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Synthesis and mu-opioid receptor affinity of a new series of nitro substituted 3,8-diazabicyclo[3.2.1]octane derivatives
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Synthesis and pharmacological activity of 4-carbamoyl-5-aryl-6-methyl-4,5-dihydropyridazin-3 (2H)-ones
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Synthesis and pharmacological activity of 4-carbamoyl-6-b-thienyl-4,5-dihydropyridazin-3-(2H) ones
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Synthesis and pharmacological activity of 4-carbamoyl-6-beta-thienyl-4,5-dihydropyridazin-3-(2H)ones
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Synthesis and pharmacological evaluation of 4,4a,5,6-tetrahydro-7,8-disubstituted-benzo[h]cinnolin-3(2H)-ones
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Synthesis and pharmacological evaluation of 4a-methyl-4,4a,5,6-tetrahydrothieno[2,3-h]cinnolin-3(2H)-ones
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Synthesis and pharmacological evaluation of 5,6-dihydrobenzo[f] cinnolin-2(3H)ones analogues of antihypertensive and antiaggregating benzo[h]cinnolinones
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Synthesis of 1-methyl -4-(N-aroyl)-piperidinamides with anti-inflammatory and analgesic activities
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Synthesis of 1-methyl-2,3-dimethyl-N(isopropyl)carbamates-4,5-dihydro-7-R'- 8-R-1H-benzo[g]indoles and evaluation of in vitro anticancer activity
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Synthesis of 3,6,7-substituted-quinoxalin-2-ones for evaluation of antimicrobial and anticancer activity. Part 2
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Synthesis of N -[ 4 (– propyl) cyclohexyl] - amides with anti – inflammatory and anlgesic activities
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Synthesis of N-[4-(Alkyl)cyclohexyl]-substituted benzamides with anti-inflammatory and analgesic activities
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Synthesis of N-[4-propyl)cyclohexyl]-amides with Anti-Inflammatory and Analgesic Activities
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Synthesis of amides with anti-inflammatory and analgesic activities
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Synthesis of amides with anti-inflammatory and analgesic activities
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Synthesis of substituted 2-ethoxycarbonyl- and 2-carboxyquinoxalin-3- ones for evaluation of antimicrobial and anticancer activity
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Synthesis, modelling, and m-opioid receptor affinity of N-3(9)-arylpropenyl-N-9(3)-propionyl-3,9-diazabicyclo[3.3.1]nonanes
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Systhesis and evaluation of gastroprotective activity of omeprazole imidazo(4,5-b) pyridine and quinoxaline 2- substituted derivatives.
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Triorganotin compounds as antimicrobial agents
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quinoxaline chemistry.Part 7. 2-[aminobenzoates]-and2-[aminobenzoylglutamate]-quinoxalines as classical antifolate agents. Sinthesis and evaluation of in vitro anticancer, anti- HIV and antifungal activity
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