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2-OXO-1,2-DIHYDROPYRIDINE-3-CARBOXAMIDE COMPOUNDS AND THEIR USE AS INHIBITORS OF PDK1 (US Patent App. 15/735,468, 2018)

Brevetto
Data di Pubblicazione:
2018
Citazione:
2-OXO-1,2-DIHYDROPYRIDINE-3-CARBOXAMIDE COMPOUNDS AND THEIR USE AS INHIBITORS OF PDK1 (US Patent App. 15/735,468, 2018) / Sestito, Simona; Daniele, Simona; Martini, Claudia; Rapposelli, Simona; Puricelli, Guido. - (2018).
Abstract:
The present invention concern a 2-oxo-1,2-dihydropyridine-3-carboxamide compound of Formula (I) and new 2-oxo-1,2-dihydropyridine-3-carboxamide compounds of Formula (II) in the treatment of pathologies which require an inhibitor of PDK1 enzyme such as diabetes, neurodegenerative diseases such as Alzheimer's and Prion Diseases, and tumours such as breast, and pancreatic cancers and glioblastoma, particularly glioblastoma.
Tipologia CRIS:
6.1 Brevetto
Elenco autori:
Sestito, Simona; Daniele, Simona; Martini, Claudia; Rapposelli, Simona; Puricelli, Guido
Link alla scheda completa:
https://iris.uniss.it/handle/11388/236198
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